DRUG in iGMDR


PD0325901PiperlongumineCYTOCHALASIN BTipifarnibNsc 632839NavitoclaxBIX01294IndisulamMerck60BMS-536924SirolimusLY 2183240IsoevodiamineKinetin ribosideFedratinibnutlin 3ParbendazoleSB225002BRD6368TozasertibQuinoclamineABT737PAC-1SelumetinibPevonedistatNSC141540NSC95397ML214ZebularineParthenolideBRD7137Fqi1GW843682XRITAGMX1778GossypolPX 12MST-312NakiterpiosinSCHEMBL2608041ImatinibBRD4770NSC23766SN-3817AAGCurcuminIdarubicinCHM-1NeopeltolideCompound 23 citrate179324-69-7DC-45-A2ItraconazoleCompound 7d-cisSepantroniumCompound 1541ATamatinibNPC26Austocystin DTriptolideSerdemetanLeucascandrolide AAvrainvillamideChaetocinBRD9876BX-795Oligomycin AISX-9Ursolic acidBRD63610PP-30Triacsin cSR-II-138AAM-580Compound 44BMS-754807ABT-751FK 866GemcitabinePI-103SalermideCompound 10b [PMID: 11504634]CD437Lovastatin acidCompound 110RotenoneChloropentafluorobenzeneBistramide ATeniposideManumycin AELCPKPemetrexed(-)-gallocatechin-3-O-gallateML 210MK-2206Tyrphostin AG-14784-methylfasudil(1S,3R)-RSL3PaclitaxelPF750QuiflaponPNU-74654FQI-2CeruleninPIK-75TanespimycinGW-405833TamoxifenNeratinibBRD4132LexibulinYK 4-279TW 37SCH-529074Cyanoquinoline 11DactolisibNVP-AUY922VorinostatJQ-1Ro 28-16752,4-dideoxy-DC-45-A2SKI IIPrima-1Brefeldin ASMR000068650Pifithrin-muOlaparibTGX-115AZD-1775PRIMA-1METBI-2536CHIR-99021DabrafenibML162VemurafenibErlotinibPluripotinBML-259BatimastatAACOCF3AfatinibCrizotinibCHEMBL1434137TrametinibCIL55ABax channel blockerPRL-3 Inhibitor ICiclosporinN9-Isopropyl-olomoucineML006PI3K pathway inhibitorVER 155008PENFLURIDOLCIL41GefitinibPDMPPLX-4720NilotinibUbistatin BImportazolePalbociclibSorafenibBRD4354LapatinibTosedostatKahalalide FSaracatinibCHEMBL399379PHA-665752MEK InhibitorSunitinibLE-135CIL56ERASTINDasatinibPurmorphamineAC55649CetuximabTAE-684TrastuzumabSparfosic acidEverolimusTivantinibSimvastatinall trans Retinoic AcidDexamethasoneOSW-1BlebbistatinPyrvinium pamoateCobimetinibPD-0325901UNC0638Tyrosine kinase inhibitorQS-11PonatinibCAY10618Pifithrin-alphamTOR inhibitorOSI-906 (Linsitinib)RefametinibCis-PlatinDocetaxelPanitumumabCapsaicinValdecoxibPK-11195RegorafenibNecrostatin-1PARP inhibitorBRAF inhibitorFatostatin AFGFR inhibitorKU0060648CI-1040BRD8958BicalutamideB02fumonisin B1TemsirolimusICL 670MitomycinCabozantinibCeritinibDoxorubicinLDN 193189ISOX DUALVismodegib (GDC-0449)MidostaurinMethotrexateCEP-701CytarabineAZD7762HSP90 inhibitorRuxolitinibCHEMBL258148BosutinibNutlin-3AKT Inhibitor VIIIObatoclaxCamptothecinCDK4/6 inhibitorFluorouracilPazopanibBleomycinGSK-461364Nutlin-3AAxitinibAZD6482AlectinibGW441756XBIRB-796BEC (hydrochloride)ElesclomolX17AAGDMOGVincaleukoblastineML203RibociclibSCHEMBL13586708BRD1812QuizartinibCeranib-2VandetanibML-030AZD-8055Gamma secretase inhibitorAvagacestat (BMS-708163)EntinostatGSK-1904529AMotesanibKo-143Nicotin-AmideHSCI1_000270NU-7441JNJ-26854165Ibrutinib (PCI-32765)BevacizumabDacomitinibBAY 61-3606ABT-263AUY922L-685458Bryostatin 1CHEMBL585951ForetinibSB-743921GSK269962AEpothilone BRucaparibBIBR-1532SB-216763BexaroteneEntrectinibPertuzumabTemozolomideTRIAZOLOTHIADIAZINEPF-562271DecitabineJAK inhibitorERK inhibitorAS601245RO-3306PD-173074ML320OSU-03012AC1NS4S0AlpelisibMEK Inhibitor (alone or in combination)JNK Inhibitor VIIIGDC-0941KU-55933PHA-793887chemotherapyBRD-K70511574GSK690693CapmatinibKW-2449ZM-447439FTI-277CX-5461Narciclasineanti-EGFR mAbsPL.DITHR1 InhibitorEGFR TK inhibitorEGFR mAb inhibitorBRD-K66453893ML311AZ628BET inhibitorCHEMBL1673039Epigallocatechin-3-monogallateEndocrine therapyGSK-650394Ado-trastuzumab emtansineMG-132EZH2 inhibitorSCHEMBL15005512OuabainLovastatinCCT007093EnzalutamideEHT-18643-Chloro-L-alanineNVP-231LSM-1215Leptomycin BCCT 018159SL 0101-1ShikoninBRD-K34222889Y-39983IPA-3Pan-RAF inhibitorOsimertinibSB590885KX2-391Omacetaxine mepesuccinateTPCA-1PF 184EmbelinCrenolanibAlisertibrTRAILrigosertibDacinostatBMS-345541StemRegenin 1KPT185NecrosulfonamideSemagacestatAICA ribonucleotideBarasertibTTNPBSarcolysinAC1MD3YPMasitinibLOXO-101SCH 79797A-770041CanertinibVeliparibMET inhibitorAR-42LBH-589CDK2 inhibitorTacedinalineLenalidomidePIK-93Vinorelbine baseDovitinibABT-888EGFR inhibitorSB525334Platinum AgentFulvestrantCarboplatinNSC74859PyrimethamineWH-4-023CGP 60474VX-702CR.1.31BWP1130SNS-032NSC87877Marinopyrrole AZM336372SNX-2112 (PF-04928473)BRD6340PLX4032QL-XI-92AZD5363S-Trityl-L-cysteineFAK inhibitorPI3K pathway inhibitor (alone or in combination)PF-573228DaporinadPembrolizumabDinaciclibI-BET151All-trans Retinoic AcidAbirateroneTGX 221Tubastatin APD318088BinimetinibErdafitinibEX-527EGFR inhibitor 1st genLetrozoleAtezolizumabFluvastatinIrinotecanPD1 Ab inhibitorX1S.3R.RSL.3MethylstatClofarabinePD153035CapecitabineTopotecanAT 7867ZINC6718453FH535DaunorubicinAlvocidibFR-180204A-443654SMO inhibitor16beta-BromoandrosteroneOSI-027BRD-K55116708PF4708671CDK2/4 inhibitorIdelalisibZSTK 474AG120ApicidinEnzastaurinHDAC inhibitorirreversible EGFR TKIsBelinostatPAK inhibitorSMER3PictilisibAZD8186STF-31anti-estrogensPlatinumBCL2 inhibitorSeliciclibX681640CP-724714BRAF inhibitors in BRAF mutant tumorIOX2RET inhibitorNSC48300ErismodegibEPZ-5676BRD-K26531177Belinostat (PXD101)BRD-K71935468IGF1R inhibitor5Z-7-OxozeaenolGSK-319347APF-3758309AURK inhibitorDBeQBRD-K35604418TretinoinGDC-0879X3.Cl.AHPCPhenforminAZD4547XAV 939PelitinibMLN 2238BrigatinibGDC-0810ABT-199 (GDC-0199)FlutamideAGK 2TivozanibLinifanibSYK inhibitorAT13387BRD-K24690302BRD-K51490254NSC19630GW2580LenvatinibPD1 blockadeNCGC00346967-01GSK-1070916STF62247LY3023414DacarbazineAG 14361CO-1686 (AVL-301)SCHEMBL618594MDM2/MDMX inhibitorspliceosome inhibitorEGFR inhibitor 3rd genPan-TRK inhibitorFumagillolCICLOPIROXInfigratinibVX-11eBRD-K92856060NintedanibAC1LE7KDMK-0752RG1084449-51-8NVP-BHG712GSK 525762ALorlatinibWEE1 inhibitorGSK2636771AZD2281PDK1 inhibitorNivolumabAmuvatinibIstradefyllineYM201636GDC-0449steroids early settingERBB2 inhibitorRAF265BRD1429BRD-K28456706WZ3105MOMELOTINIBAS 605240DNA-PKc inhibitorARN-509LomeguatribSU 11274CCT036477SRT-1720SRC inhibitorZ-LLNle-CHOAG-221KHS101ML239HLI-373Zibotentan (ZD4054)TegafurPhloretinNelarabineCD1530ALK inhibitorNVP-ADW742VNLG/124BRD-K94991378WZ 4002AZD1480MetforminAbemaciclibSJ-172550AZ3146BirinapantEPZ-6438JW-7-52-1ProchlorperazineTHZ-2-102-1MPS1-IN-1BX 912CDK9 InhibitorOxaliplatinFMKQW-BI-011MercaptopurineBRD-A86708339OSI-930BRD-K97651142mTORC1/2 inhibitorBMN 673ChlorambucilHC-067047ThioguanineMGCD-265TL-2-105NG25BMS-509744PFI-1SB-715992BRD-A71883111SGC0946ML050Tankyrase inhibitorWHI-P97CMKCP466722GNF-2JW-7-24-1LRRK2-IN-1CediranibHG6-64-1AZD6738TAK-788QL-XII-61FingolimodKIN001-236allosteric AKT inhibitorBRD-K66532283GSK429286AAT-406EX-8678Bardoxolone methylJQ12BRD-K02251932RO4987655XMD13-2PP-242Hormone TherapyCGP-082996ML029GSK-3 Inhibitor IXWZ8040BIX02189AVICIN DTL-1-85irreversible EGFR T790M inhibitorPD-1 InhibitorXMD15-27Trastuzumab EmtansineBRD-K61166597CDK4 inhibitorMdivi-1XL765EGFR inhibitor 2nd genSGX-523TG100-115NimotuzumabCID 5951923TAK-715BRD-K13999467TandutinibQL-X-138BI-D1870CAY10603BRD1835PI3K alpha inhibitorMI-2BRD-K93923542-001-01-9TaselisibCOL-3THZ-2-49R428HSP90 inhibitor (in combination)BRD-K17060750AT-7519MyricetinPF-03084014FLT3 inhibitorBRD-K63431240EPZ005687PLX3397RO4929097Sym00417-DMAGPKC inhibitorKU-60019AzacitidineCH 55PF 4800567 HydrochlorideArsenic TrioxideIsonicotinohydroxamic acidRepligen-136Genentech Cpd 10KU0063794BRD-A94377914novel ALK inhibitorCompound 1bX16 beta bromoandrosteroneHBX-41108MEK Inhibitor +/- PI3K pathway inhibitorMDM2 inhibitorPomalidomideBleomycin a2BRD55319MI.1Porcupine inhibitor844499-71-4GANT61CUDC-101ETP-46464CyclophosphamidePyrazolanthroneTubulin inhibitorBRD-K41597374UNC-0321LestaurtinibGSK2141795 (hydrochloride)Pramlintide [USAN]BRD-K45681478FAS inhibitorUNC1215RidaforolimusSB-505124SilmitasertibDOT1L inhibitorArabinosylguanine6-MercaptopurineBRD-M00053801Cucurbitacin ILY-294002BRD9647QL-VIII-58Aromatase ihibitorEZH2 inhibitor in RAS wtNSC-207895COT Inhibitor-2BRD-K52037352BRD-K09344309first-generation and irreversible EGFR TKIsNVP-BSK805IDH1 inhibitorHG-5-88-01PF-543SCHEMBL2593705BrivanibBRD8899T091317AR antagonistE-3810BCL.LZH.4AndrogenSotrastaurin6-ThioguaninePIK3CA inhibitorPerifosineATR inhibitorML031MyriocinTaxaneAZD-9291MTX sodiumR1507chemotherapy (HER2 ampl)TrifluoperazineSpautin-1BRD-K85133207MEK Inhibitor/anti-EGFR mAbAdoptive T-cell TransferLY2157299KIT inhibitorBCL-XL inhibitornovel MEK inhibitorHydroxy VandetanibBH3novel estrogen receptor degraderAGI-5198JAK/TBK1/IKK? inhibitorElocalcitolBRD-K14844214GSK4112anti-tubulin agentsThalidomidenon-allosteric AKT inhibitoranti-HER3 mAbsMDM2 inhibitor (tumors TP53 wt)IPI-504SLC44A4 inhibitornovel anti-EGFR mAbsJAK inhibitor (alone or in combination)CDK7 inhibitorATM inhibitorPIK3CB inhibitorBET inhibitors in LKB1 wtCDK6 inhibitorOctreotideIC-87114GSK 1059615AspirinBRD-K09587429BRD-K29086754BMS614LHRH analogues or antagonistKH-CB19VALPROIC ACIDBRD-A05715709ApitolisibLevoleucovorinIDH2 inhibitorIpilimumabBRD4 inhibitorARRY-470PDL1 inhibitorERBB3 mAb inhibitorMEDI0680MLN2480EPHA3 inhibitorCDK4/CDK6 inhibitor (abemaciclib)SB-431542BRD-K96970199PandacostatPIM inhibitor138402-11-62,4-PyrimidinediamineHM61713NSC348884AmrubicinAdjuvant ChemotherapyMLL1 inhibitorCH5132799mTOR kinase inhibitorMEDI4736RapaLink-1BRD-K02492147BRD-K78574327next-generation AR antagonistsBRD-K99006945BGB659AV-203Antiangiogenic TherapyOMP-52M51AR inhibitor next genVEGFR inhibitornovel FLT3 inhibitorAZD7545ML258AZD3463Kinome_3629eribulinOMP-59R5StaurosporineML334 diastereomerVolasertibAnthracyclineSZ4TA2Skepinone-LPDGFR inhibitorQL-XII-47SU-5614HG-5-113-01ILORASERTIBVorapaxarRadioiodine Uptake TherapyPI3K/MEK inhibitorTazemetostatNOTCH1 AntibodyBRD-K37390332BRD-K84807411Spliceostatin ARindopepimutXL-647BRD-K88742110SteroidCixutumumabSCH772984BRD-K29313308Anti-CD33OICR-9429AZ909TRK inhibitorCTLA4 inhibitorBRD-K48477130CI-976HyperforinSRC inhibitor (in combination with PI3K/MEK inhibitors)Trichostatin AIPR-456Betulinic acidBRD-K19103580AEE788StatticXMD11-85hAnti-ERBB3 AgentsC20H13BrN2O3S2ProcarbazineSAR405838MocetinostatMEK Inhibitor enhanced radioiodine uptake852475-26-4XMD 8-921166227-08-2HER2 inhibitorAnastrozoleNilutamideCbl0137IMGENEXPilaralisibGDCVTX-11eDirigestranAlemtuzumabDS-3032BTIM-3 InhibitorMEK Inhibitor in EGFR mutantKetoconazoleRadiationIMO2-(1H-Indazol-4-yl)-6-(4-methanesulfonylpiperazin-1-ylmethyl)-4-morpholin-4-yl-thieno[3,2-d]pyrimidineIRAK-1/4 InhibitorTacrolimusmTOR inhibitor (in SH2B3 deleted)BPTESFolfox protocolInduction TherapyCHK1/2 inhibitorVemurafenib and panitumumab (in BRAF V600E mutated)IGF1R antibodiesSB-202190CBB1007GNE-617CabazitaxelSR1001PSEUDOEPHEDRINEall trans Retinoic Acid (non-FLT3 ITD AML)PYR-41MLS006011051G007-LKBCR-ABL1 inhibitorsBRD-K64610608ARS-85317224927anti-CTLA4 mAbsPan-TK inhibitorAminoglutethimideFACT inhibitorBRD-K49290616LonafarnibBuparlisibIpatasertibBRD-K33514849PatritumabBRD-K50799972U0126IGF1R Monoclonal AntibodyIrinotecan plus CHK1/2 inhibitor in ATM deficient tumorBRD-K16147474GDC-0623Crizotinib and vemurafenib (in BRAF V600E mutated)4-HydroxytestosteroneEpirubicinTrastuzumab-based chemotherapyCisplatin-4-methylpyridineAspirin in adjuvant settingAvelumab4-HydroxytamoxifenGanetespib (STA-9090)IU1TAK-733JW 55CDK4 inhibitor (tumors with RB expression)CimetidineGSK321OrteronelFGIN-1-27Necrostatin-7Savolitinib9F7-F11Farnesylthiosalicylic acidBMS-270394Monomethyl auristatin ESU-5402Bendamustine HClBRD-K30748066PI3K InhibitorCarmustineBRD-K04800985Cyproterone AcetateKi8751Ethyl L-asparaginateBRD-K90370028RaltitrexedBRD-K48334597MEK Inhibitor in BRAF mutant tumorsSildenafilCc-223PI3K beta inhibitorJW74O(6)-benzylguanineTrastuzumab in HER2-amplifiedSalinomycinFasudilRG7356AZD-5438ACLY SiRNAWYE-354ESR1 inhibitorSaridegib (USAN)SGK1 inhibitorBRD-K44224150BRD-K41334119EGFR TK inhibitor (EGFR mut disease)ATP-competitive AKT inhibitorsselective FGFR inhibitorTrastuzumab (ANXA1 high)Trastuzumab-based therapyGSK-J4ConatumumabAmilorideFSC-231CAY-10594C6 ceramideNeratinib plus temsirolimusFOLFIRI regimenMLN0128LY3009120OmipalisibTrastuzumab (in HER2 co-amplified)JAK3 Inhibitor IIETOMOXIRAG-1296X968Trametinib (plus imatinib in BCR-ABL)SitagliptinLGK974G-573BRD-K33199242(R)-VerapamilJNK-IN-2OnartuzumabAnti-CD123Trastuzumab in HER2-amplFlavopiridolLomustine