DSTYK


Summary: This gene encodes a dual serine/threonine and tyrosine protein kinase which is expressed in multiple tissues. It is thought to function as a regulator of cell death. Multiple transcript variants encoding different isoforms have been found for this gene. [provided by RefSeq, Dec 2008].

NameOMIM IDEnsembl IDHGNC IDPHARMGKB IDMap Location
dual serine/threonine and tyrosine protein kinaseMIM:612666Ensembl:ENSG00000133059HGNC:HGNC:29043PA1647188611q32.1

GO terms in DSTYK


Term TypeEvidence TypeGO Term IDGO Des.
CCIDAGO:0005737cytoplasm
CCIDAGO:0016323basolateral plasma membrane
CCIDAGO:0016324apical plasma membrane
CCIEAGO:0030054cell junction
BPIEAGO:0018108peptidyl-tyrosine phosphorylation
BPIMPGO:0033674positive regulation of kinase activity
BPIMPGO:0043066negative regulation of apoptotic process
BPIDAGO:0044344cellular response to fibroblast growth factor stimulus
BPIMPGO:0045743positive regulation of fibroblast growth factor receptor signaling pathway
BPIMPGO:0070374positive regulation of ERK1 and ERK2 cascade
MFIEAGO:0004712protein serine/threonine/tyrosine kinase activity
MFIEAGO:0004713protein tyrosine kinase activity
MFIEAGO:0005524ATP binding

Gene expression in normal tissue: DSTYK

Gene-model tissue-cancer distribution: Bubble Plot

Gene-drug pathway distribution

Pathways in DSTYK


DatabasePathway IDPathway Des.

Gene-Drug: Aster Plot


Drug IDDrug NameModel Num.
iGMDRD505Pevonedistat2
iGMDRD263AACOCF36
iGMDRD246NPC263
iGMDRD82Quiflapon4
iGMDRD367Ro 28-16752
iGMDRD871BRD63683
iGMDRD286Nsc 6328393
iGMDRD882CIL413
iGMDRD662JQ-13
iGMDRD221Tamoxifen5
iGMDRD705Nakiterpiosin3
iGMDRD6AM-5806
iGMDRD192CIL564
iGMDRD77Itraconazole3
iGMDRD267Oligomycin A3
iGMDRD137Indisulam3
iGMDRD901ELCPK5
iGMDRD132(-)-gallocatechin-3-O-gallate1
iGMDRD883CIL55A6
iGMDRD499PDMP2
iGMDRD345Compound 10b [PMID: 11504634]2
iGMDRD522ML-0301
iGMDRD405PIK-753
iGMDRD307Manumycin A4
iGMDRD486Tosedostat2
iGMDRD584VER 1550081
iGMDRD512nutlin 33
iGMDRD640CAY106181
iGMDRD64Parbendazole1
iGMDRD874BRD89583
iGMDRD23Gossypol4
iGMDRD562Navitoclax1
iGMDRD780PP-303
iGMDRD782DC-45-A22
iGMDRD226ML0063
iGMDRD318PAC-13
iGMDRD52Rotenone1
iGMDRD394BX-7953
iGMDRD375GW-4058333
iGMDRD201SKI II1
iGMDRD193Fqi11
iGMDRD779PRL-3 Inhibitor I3
iGMDRD546BMS-7548073
iGMDRD483SCH-5290743
iGMDRD126Tipifarnib1
iGMDRD599Salermide3
iGMDRD889Compound 7d-cis3
iGMDRD579PF7502

Gene in drug-gene network: Network Plot

Gene-drug targets distribution

Gene Structure: PDB

Models in DSTYK

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