iGMDRD260
| Standard Name | CHEMBL | Pubchem CID | Drug Status | Drug Type |
|---|---|---|---|---|
| FQI-2 | CHEMBL3608990 | 5172540 | Alone | Small Molecule |
Drug-model tissue-cancer distribution: Bubble Plot
Drug-gene pathway enrichments
Drug-gene GO enrichments
Drug-Gene: Aster Plot
| Gene ID | Gene Name | Model Num. |
|---|---|---|
| 1105 | CHD1 | 2 |
| 27125 | AFF4 | 3 |
| 7514 | XPO1 | 1 |
| 8999 | CDKL2 | 2 |
| 5296 | PIK3R2 | 2 |
| 5027 | P2RX7 | 1 |
| 23085 | ERC1 | 2 |
| 5261 | PHKG2 | 2 |
| 7750 | ZMYM2 | 1 |
| 4926 | NUMA1 | 2 |
| 11183 | MAP4K5 | 1 |
| 4627 | MYH9 | 1 |
| 2956 | MSH6 | 4 |
| 2200 | FBN1 | 3 |
| 9706 | ULK2 | 3 |
| 347365 | ITIH6 | 2 |
| 3845 | KRAS | 1 |
| 55215 | FANCI | 1 |
| 8289 | ARID1A | 2 |
| 2335 | FN1 | 3 |
| 84700 | MYO18B | 5 |
| 2475 | MTOR | 4 |
| 9475 | ROCK2 | 1 |
| 8780 | RIOK3 | 1 |
| 7764 | ZNF217 | 3 |
| 10395 | DLC1 | 1 |
| 5133 | PDCD1 | 6 |
| 11116 | FGFR1OP | 3 |
| 390502 | SERPINA2 | 2 |
| 64783 | RBM15 | 4 |
| 10892 | MALT1 | 1 |
| 4170 | MCL1 | 1 |
| 3066 | HDAC2 | 3 |
| 10142 | AKAP9 | 2 |
| 23310 | NCAPD3 | 1 |
| 6732 | SRPK1 | 1 |
| 1404 | HAPLN1 | 4 |
| 7048 | TGFBR2 | 3 |
| 51199 | NIN | 1 |
| 1387 | CREBBP | 4 |
| 2043 | EPHA4 | 2 |
| 1859 | DYRK1A | 1 |
| 2313 | FLI1 | 3 |
| 5579 | PRKCB | 2 |
| 31 | ACACA | 1 |
| 10178 | TENM1 | 1 |
| 51755 | CDK12 | 4 |
| 79858 | NEK11 | 1 |
| 8295 | TRRAP | 4 |
| 10438 | C1D | 5 |
| 5159 | PDGFRB | 1 |
| 7373 | COL14A1 | 1 |
| 145264 | SERPINA12 | 3 |
| 2033 | EP300 | 4 |
| 64324 | NSD1 | 3 |
| 55728 | N4BP2 | 4 |
| 54477 | PLEKHA5 | 2 |
| 57670 | KIAA1549 | 4 |
| 22861 | NLRP1 | 2 |
| 440279 | UNC13C | 3 |
| 2115 | ETV1 | 1 |
| 4301 | AFDN | 1 |
| 84033 | OBSCN | 3 |
| 1540 | CYLD | 1 |
| 10342 | TFG | 3 |
| 22984 | PDCD11 | 2 |
| 6091 | ROBO1 | 6 |
| 2042 | EPHA3 | 6 |
| 2260 | FGFR1 | 3 |
| 116986 | AGAP2 | 2 |
| 83990 | BRIP1 | 3 |
| 284217 | LAMA1 | 4 |
| 269 | AMHR2 | 1 |
| 55681 | SCYL2 | 1 |
| 65266 | WNK4 | 2 |
| 8643 | PTCH2 | 2 |
| 65217 | PCDH15 | 1 |
| 79971 | WLS | 5 |
| 286826 | LIN9 | 3 |
| 23191 | CYFIP1 | 1 |
| 9759 | HDAC4 | 1 |
| 6709 | SPTAN1 | 3 |
| 8215 | DVL1P1 | 1 |
| 6793 | STK10 | 3 |
| 9472 | AKAP6 | 1 |
| 2778 | GNAS | 1 |
| 80243 | PREX2 | 5 |
| 139285 | AMER1 | 2 |
| 575 | ADGRB1 | 1 |
| 5924 | RASGRF2 | 3 |
| 9564 | BCAR1 | 2 |
| 1496 | CTNNA2 | 5 |
| 2066 | ERBB4 | 3 |
| 10413 | YAP1 | 3 |
| 2201 | FBN2 | 2 |
| 1029 | CDKN2A | 1 |
| 57523 | NYNRIN | 3 |
| 5834 | PYGB | 1 |
| 58508 | KMT2C | 6 |
| 2099 | ESR1 | 1 |
| 6092 | ROBO2 | 1 |
| 4855 | NOTCH4 | 3 |
| 25836 | NIPBL | 6 |
| 3791 | KDR | 1 |
| 4292 | MLH1 | 3 |
| 114788 | CSMD3 | 1 |
| 2263 | FGFR2 | 3 |
| 4086 | SMAD1 | 1 |
| 1019 | CDK4 | 3 |
| 55034 | MOCOS | 3 |
| 23043 | TNIK | 3 |
| 7038 | TG | 3 |
| 55589 | BMP2K | 3 |
| 65125 | WNK1 | 1 |
| 7175 | TPR | 3 |
| 5871 | MAP4K2 | 3 |
| 80205 | CHD9 | 3 |
| 8997 | KALRN | 3 |
| 23269 | MGA | 5 |
| 23469 | PHF3 | 5 |
| 4089 | SMAD4 | 3 |
| 6654 | SOS1 | 3 |
| 546 | ATRX | 1 |
| 51366 | UBR5 | 3 |
| 23678 | SGK3 | 2 |
| 54756 | IL17RD | 1 |
| 1978 | EIF4EBP1 | 1 |
| 57144 | PAK5 | 1 |
| 4214 | MAP3K1 | 8 |
| 3702 | ITK | 5 |
| 440275 | EIF2AK4 | 3 |
| 3239 | HOXD13 | 4 |
| 3720 | JARID2 | 2 |
| 1687 | GSDME | 1 |
| 2318 | FLNC | 1 |
| 10565 | ARFGEF1 | 2 |
| 64919 | BCL11B | 4 |
| 675 | BRCA2 | 7 |
| 26166 | RGS22 | 1 |
| 607 | BCL9 | 4 |
| 7075 | TIE1 | 2 |
| 640 | BLK | 1 |
| 11064 | CNTRL | 3 |
| 2624 | GATA2 | 3 |
| 5789 | PTPRD | 1 |
| 8021 | NUP214 | 2 |
| 10461 | MERTK | 1 |
| 26278 | SACS | 2 |
| 833 | CARS | 1 |
| 7917 | BAG6 | 2 |
| 375056 | MIA3 | 3 |
| 91754 | NEK9 | 3 |
| 93627 | TBCK | 2 |
| 7153 | TOP2A | 3 |
| 57082 | KNL1 | 4 |
| 1981 | EIF4G1 | 5 |
| 22976 | PAXIP1 | 3 |
| 23532 | PRAME | 1 |
| 4863 | NPAT | 2 |
| 780 | DDR1 | 3 |
| 339345 | NANOS2 | 2 |
| 120892 | LRRK2 | 2 |
| 5205 | ATP8B1 | 2 |
| 9321 | TRIP11 | 2 |
| 9451 | EIF2AK3 | 3 |
| 8491 | MAP4K3 | 1 |
| 4853 | NOTCH2 | 3 |
| 23049 | SMG1 | 1 |
| 10752 | CHL1 | 3 |
| 667 | DST | 6 |
| 23281 | MTUS2 | 3 |
| 115701 | ALPK2 | 4 |
| 6770 | STAR | 3 |
| 7273 | TTN | 4 |
| 23389 | MED13L | 2 |
| 55561 | CDC42BPG | 3 |
| 22843 | PPM1E | 3 |
| 344905 | ATP13A5 | 3 |
| 4297 | KMT2A | 1 |
| 7248 | TSC1 | 3 |
| 4619 | MYH1 | 1 |
| 57680 | CHD8 | 1 |
| 2317 | FLNB | 2 |
| 10111 | RAD50 | 5 |
| 9659 | PDE4DIP | 6 |
| 6093 | ROCK1 | 1 |
| 5927 | KDM5A | 5 |
| 5587 | PRKD1 | 6 |
| 5589 | PRKCSH | 4 |
| 57448 | BIRC6 | 4 |
| 2131 | EXT1 | 3 |
| 3717 | JAK2 | 3 |
| 23139 | MAST2 | 2 |
| 2157 | F8 | 2 |
| 5506 | PPP1R3A | 2 |
| 6778 | STAT6 | 2 |
| 1030 | CDKN2B | 1 |
| 3977 | LIFR | 3 |
| 5894 | RAF1 | 1 |
| 182 | JAG1 | 3 |
| 2122 | MECOM | 3 |
| 5925 | RB1 | 1 |
| 1515 | CTSV | 2 |
| 2065 | ERBB3 | 1 |
| 4638 | MYLK | 1 |
| 7040 | TGFB1 | 3 |
| 30849 | PIK3R4 | 2 |
| 9878 | TOX4 | 1 |
| 142 | PARP1 | 3 |
| 2261 | FGFR3 | 3 |
| 2073 | ERCC5 | 3 |
| 55422 | ZNF331 | 2 |
| 3092 | HIP1 | 2 |
| 4763 | NF1 | 2 |
| 55791 | LRIF1 | 4 |
| 4193 | MDM2 | 2 |
| 2178 | FANCE | 2 |
| 1499 | CTNNB1 | 4 |
| 2892 | GRIA3 | 3 |
| 4486 | MST1R | 3 |
Gene in drug-gene network: Network Plot
Models in FQI-2

